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Publication

The Strecker reaction coupled to Viedma ripening: a simple route to highly hindered enantiomerically pure amino acids

Article
Chem. Comm., 2018, 54, 10832-10834
Year
2018
Customer
AMOLF
Site
Department
MCS people
Michel Leeman, Richard Kellogg
Publication

Charting Biologically Relevant Spirocyclic Compound Space

Article
Chem. Eur. J. 2017, 23 (3), 703-710
Year
2017
Customer
ELF
Site
Department
MCS people
Gerhard Müller, Tim Berkenbosch, Jorg Benningshof
Publication

Design and Synthesis of Enantiomerically Pure Decahydroquinoxalines as Potent and Selective k-Opioid Receptor Agonists with Anti-Inflammatory Activity in Vivo

Article
J. Med. Chem. 2017, 60 (6), 2526-2551
Year
2017
Customer
Dr. August Wolff
Site
Department
MCS people
Peter Molenveld, Roy Storcken, Renaud Bouzanne des Mazery, Geert-Jan Sterk, Reshma Autar, Marjon Bolster, Clemens Wagner, Frank van Holst, Anita Wegert
Publication

Discovery, Structure-Activity Relationship, and Binding Mode of an Imidazo[1,2-a]pyridine Series of Autotaxin Inhibitors

Article
J. Med. Chem. 2017, 60 (17), 7371-7392
Year
2017
Customer
Galapagos
Site
Department
MCS people
Jörg Heiermann, Willem Hengelveld, Gregor Pilzak
Publication

Piperidine and octahydropyrano[3,4-c] pyridine scaffolds for drug-like molecular libraries of the European Lead Factory

Article
Bioorg. Med. Chem. 2017, 5160 - 5170
Year
2017
Customer
Leiden Institute of Chemistry
Site
Department
MCS people
Dirk Vandenput, Joeri Scheidt, Jorg Benningshof
Publication

Synthesis and Properties of 2-Oxa-6-azaspiro[3.3]heptane Sulfonate Salts

Article
Synthesis 2017, 49 (11), 2394-2401
Year
2017
Customer
Bayer Pharma
Site
Department
MCS people
Richard van der Haas, Jeroen Dekker, Eric Damen
Publication

Efficient reagent-saving method for the N-terminal labeling of bioactive peptides with organometallic carboxylic acids by solid-phase synthesis

Article
Organometallics (2016), 35(18), 3192-3196
Year
2016
Customer
Wageningen University
Site
Department
MCS people
Jack Slootweg
Publication

Securing Important Strigolactone Key Structures: Orobanchol and 5-Deoxystrigol

Article
Eur. J. Org. Chem. 2016 (12), 2163–2169
Year
2016
Customer
Radboud University
Site
Department
MCS people
Colinda van Tilburg‐Joukema, Bram van Oss, Peter Molenveld
Publication

Strategic and tactical approaches to the synthesis of 5,6-dihydro-[1,2,4]oxadiazines

Article
Heterocycles 2016, 92 (12), 2166-2200.
Year
2016
Customer
Mercachem
Site
Department
MCS people
Johan Veerman, Yorik Bruseker, Bart van Esseveldt, Erik Heijne, Tommi Meulemans, Peter van Rijnsbergen, Wim Zonneveld
Publication

Synthesis and evaluation of analogs of the phenylpyridazinone NPD-001 as potent trypanosomal TbrPDEB1 phosphodiesterase inhibitors and in vitro trypanocidal

Article
Bioorg. Med. Chem. 2016, 24 (7), 1573-1581
Year
2016
Customer
VU
Site
Department
MCS people
Johan Veerman, Toine van den Bergh, Geert-Jan Sterk

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